4-aminopyridine 4-AP 5-HT 5-HT transporter 5-HT1 5-HT2 5-HT3 5-HT4 5-HT5 5-HT6 5-HT7 5-hydroxytryptamine 7-chlorokynurenic acid accommodation ACE inhibitor acebutolol acetaldehyde dehydrogenase acetic acid acetylcholine acetylcholineesterase ACh AChE ACTH adenosine adenosine-diphosphate adenosine-triphosphate adenylyl cyclase ADP adrenal cortex adrenal medulla AF-DX 116 afterhyperpolarization agonist AHP alanine albuterol alcohol alcohol dehydrogenase aldehyde aldosterone allosteric alloxazine alpha receptors alpha-bungarotoxin alpha-methyl-5-hydroxytryptamine alpha-methyl-para-tyrosine alpha-methyldopa alpha-subunit alpha1 receptor alpha2 receptor alternative splicing ambenonium amino acid amino-terminal (NH2) amitriptyline AMPA receptor amphetamines androgen anion anomolous rectifier antagonist antihypertensive antipsychotics AP4 AP5 apamin APE APV aqueous arachadonic acid arecoline aspartic acid (aspartate) asthma atenolol ATP atropine autoreceptor AVP baclofen barbiturate BAY-K-8644 benzodiazepine beta receptors beta-amyloid peptides beta-cells beta-endorphin estradiol beta-subunit beta1 receptor beta2 receptor beta3 receptor bethanechol bicuculline binding binding site biosynthetic enzyme BK channel blood pressure blood-brain barrier Bmax botulinum toxin (botulism) bound bradykinin bretylium bromocriptine bufotenin bupropion butoxamine Ca2+ Ca2+-ATPase CACA caffeine calbindin calcineurin calcitonin calcium binding proteins calcium currents calcium ions calcium spike calcium stores calcium-calmodulin dependent kinase II calcium-dependent Ca2+ release calcium-dependent K+ currents calmodulin CAM-KII cAMP capsaicin carbachol carbidopa carboxy-terminal (COOH) cascade catalytic subunit catecholamines cation CCK cerebrospinal fluid cGMP channel charge gradient charybdotoxin chloride current chloride ion chlorotoxin chlorpromazine cholera toxin choline cirazoline Cl- clearance rate clonidine clorgyline clozapine CNQX coagonist cocaine codeine cofactor compartment competition competitive antagonist COMT concentration curve concentration gradient corticosteroids corticotropin-releasing factors cortisol coupling CPA CPP CPT CPX CREB CRF cross-linked CSF curare current-clamp current-voltage relationship cyclic AMP cyclic GMP cyclic nucleotide -phosphodiesterase cyclopropane cyprodime cytochrome P450 D-cycloserine d-tubocurarine D1 receptor D2 receptor D3 receptor D4 receptor D5 receptor DA DA transporter DAG DAMGO DARRP-32 DCS decamethonium degradatory enzyme delayed rectifier delta receptor deltramethin dendrotoxin depolarization depolarization block deprenyl desipramine dexamethasone diacylglycerol diazepam (valium) diethyl ether digitalis dihydromorphine dihydropyridine dihydroxyphenylalanine diltiazem dimer disinhibition disulfiram divalent DMPP DMT DNQX dobutamine domoic acid (domoate) dopamine dopamine-beta-hydroxylase dose-response curve down-regulation drug dynorphin A EC50 ED50 eicosanoids electrostatic gradient endocytosis enflurane enhancement enzyme ephedrine epinephrine EPSC EPSP esmolol estrogen ethanol etorphine excitotoxicity exocytosis exocytoxin extracellular facilitation false transmitters fluoxetine fluphenazine fluvoxamine free full agonist G-protein GABAA receptor GABAB receptor GABAC receptor GAD gallamine ganglion ganglionic blocker gating GDP general anesthetic Gi glia glucocorticoid glucose glutamate decarboxylase glutamic acid (glutamate) glutaminase glycine glycine site glycolysis Go Gs GTP GTP-gamma-S guanabenz guanethidine guanine-diphosphate guanine-triphosphate H1 receptor H2 receptor HA-966 half-life half-time haloperidol halothane heart rate hemicholinium heroin hexamethonium Hill coefficient Hill plot himbacine histamine histidine homo-cysteic acid hormone hydrocortisone hydrophilic hydrophobic hydrophobicity plots hypertension HPA axis I Ca2+ I cl- I K+ I/V curve IM imipramine INa+ inactive indoleamines inhibitor insecticide insoluble insulin intracellular intracellular free Ca2+ ion channel ionic gradient ionophore ionotropic IP3 IP3 receptor IPSC IPSP isamoltane isoflurane isoguvacine isopropanol isoproterenol K+ kainate receptor kainic acid (kainate) kappa receptor kappa-bungarotoxin KD kinase kinetics kitanserin L-type channel labetalol LADME LD50 leu-enkephalin lidocaine ligand ligand-gated channel ligand-receptor complex lipophilic lobeline local anesthetic LSD-25 lysergic acid diethylamide M-current M1 M2 M3 M4 M5 malathion MAO MAO-A MAO-B MAP-2 mecamylamine melatonin mescaline mesulergine met-enkephalin metabolism metabotropic receptor methacholine methadone methamphetamine methanol methoxamine methoxyflurane methylatropine methylcarbamylcholine methylphenidate metoclopramide metoprolol Mg2+ mGLUr mineralocorticoid mitochondria MK-801 MMDA modulatory monoamine oxidase monoamine oxidase inhibitor monomer monovalent morphine mu receptor muscarine muscarinic muscimol N-type channel Na+ Na+/K+-ATPase nadolol nalorphine naloxone naltrexone naltrindole NBQX NE NE transporter nefazodone neostigmine nerve gas neuroleptics neuromodulatory neuromuscular junction neuropeptidases neuropeptide Y neurotensin neurotransmitter release nicotine nicotinic nifedipine nimodipine nipecotic acid nitrous oxide nitrous oxide synthase NO noncompetitive antagonist nonhydrolyzable-GTP nonspecific nonvesicular relesase noradrenaline norepinephrine nortriptyline obidoxime okadaic acid omega-agatoxin omega-conotoxin opiates ouabain oxazepam oxidative metabolism oxotremorine oxymorphone oxytocin P-type channel P2 receptor paired pulse depression papaverine paraoxon parathion pargyline paroxetine partial agonist PCP PDE pentazocine pentobarbital pergolide permeability pertussis toxin pH phaclofen phencyclidine phenelzine phenmetrazine phenothiazines phenoxybenzamine phentolamine phenylephrine phenylzine phenytoin phosphatase phosphatidylinositol phosphodiesterase phospholipase A phospholipase C phospholipase D phosphorylation physostigmine picrotoxin pilocarpine pimozide pindolol PIP2 pirenzepine PKA pKa PKC PLA placebo plasma protein bound PLC PLD pore postganglionic postsynaptic potassium current potassium ion pralidoxime prazosin precursor prednisone preganglionic pregnenolone presynaptic procaine procaterol product progesterone promoter regions proopiomelanocortin propanolol protein kinase A protein kinase C protein phosphatase I protein phosphatase II prozac psilocybin pump purinergic purinoceptor pyrethrin pyrethroids Q-type channel quanta quisqualic acid (quisqualate) QX-314 raclopride receptor receptor occupancy receptor proliferation receptor turnover regulatory protein phosphatase regulatory subunits reluctance remoxipride reserpine residue reuptake inhibitors reverse agonist risperidone rough endoplasmic reticulum routes of administration: a. im b. iv c. ip d. icv e. oral f. sublingual R-PIA ryanodine ryanodine receptor saclofen sarin saturable saturation saxitoxin Scatchard plot Schild plot scopolamine second messenger sedation sensitization serine serotonin sertraline sigma receptor single-channel recording SK channel sodium current sodium ion sodium-potassium pump soluble soman specific spine spiperone spiroperidol steroids strychnine-insensitive strychnine-sensitive subconductance state substance P substrate subunit succinylcholine sufentanyl fentanyl suicide antagonist sumatriptan T-type channel tachycardia tacrine taurine TEA telenzepine testosterone tetanus toxin tetraethylammonium tetramethylammonium thapsigargin thorazine timolol TMA tolerance toxin trans-(1S,3R)-ACPD transmembrane transporter trazodone tricyclic antidepressants trifluoperazine trimer trimethaphan trimipramine tropicamide tryptamine tryptophan tryptophan hydroxylase TTX tyrosine tyrosine hydroxylase unbound up-regulation uptake inhibitor vasodilation vasodilator vasopressin verapamil vesamicol vesicle vesicular relesase voltage-dependent channel voltage-gated channel yohimbine zacopride